Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_02704
Ion Channel
Potassium voltage-gated channel subfamily A member 5
Peptide Function
Blocker
Gene Name
KCNA5
Activity Data (nM)
IC50
460 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
YCQKWMWTCDSERKCCEGMVCRLWCKKKLW
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Not available
Peptide Species
Thrixopelma pruriens (Peruvian green velvet tarantula)
Peptide Name
Beta/omega-theraphotoxin-Tp2a
CAS Number
484598-36-9
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−80 mV
Temperature
20–22 °C
Test Method
Patch-clamping
Test Species
HEK293 cell (Homo sapiens embryonic kidney 293 cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available